| Description |
1 online resource |
| Series |
Biochemistry research trends |
|
Biochemistry research trends series.
|
| Contents |
BIOACTIVE HETEROCYCLES: SYNTHESIS AND BIOLOGICAL EVALUATION; BIOACTIVE HETEROCYCLES: SYNTHESIS AND BIOLOGICAL EVALUATION; Library of Congress Cataloging-in-Publication Data; Contents; Preface; About the Editors; Contributors; Chapter 1: Multipotent 1,8-Naphthyridines, as New Tacrine Analogues, for the Treatment of Alzheimer's Disease; Abstract; 1. Introduction; 2. 4H-Pyrano [2,3-b]Pyridines (Pyranotacrines); 2.1. Synthesis; 2.2. Pharmacology; 3. Furo and Thieno[2,3-b]pyridines (Furo and Thienotacrines); 3.1. Synthesis; 4. 4-Aryl-1,8-naphthyrydines (Pyridotacrines); 4.1. Synthesis |
|
4.2. PharmacologyConclusion; References; Chapter 2: Pyrrolo [1,2-a] Quinolines: Synthesis and Biological Activity; Abstract; 1. Introduction; 2. Synthetic Routes to Pyrrolo[1,2-a]Quinolines; 2.1. Synthesis Starting from Quinoline and Its Derivatives; 2.2. Synthesis Starting from Pyrroles; 2.3. Other Methods for Obtaining Pyrrolo[1,2-a]Quinolines; 2.4. Bioactive Compounds Based on Pyrrolo[1,2-a]Quinolines; Conclusion; Acknowledgments; References; Chapter 3: Aziridines: Synthesis and Bioactivity; Abstract; 1. Introduction; 2. Overview and General Features; 3. Synthesis of Aziridines |
|
3.1. From Addition to Alkenes3.2. From Ü, Ý-Unsaturated Carbonyl Compounds; 3.3. From Imines; 3.4. From Ring Closure of Haloamines and Amino Alcohols; 3.5. By Ring Transformation of Epoxides; 3.6. Miscellaneous Synthesis; 4. Biological Activity of Aziridines; 4.1. Cytotoxic and Anticancer Activities; 4.2. Antimicrobial Activities; 4.3. Protein Inhibitor Aziridines; 4.4. Antibiotic and Miscellaneous Activities of Aziridines; Conclusion; References; Chapter 4: Bioactivity and Synthesis of Substituted Imidazole Motifs; Abstract; 1. Introduction |
|
2. Biological Importance of Substituted Imidazole Derivatives2.1. Cyclooxygenase-2 (COX-2) Inhibitors Activity of imidazoles; 2.2. Inhibitors of p38 MAP Kinase Activity of imidazoles; 2.3. Combretastatin A-4 (CA-4) Analogues with Antitumor Activity; 2.4. Modulators of P-glycoprotein (P-gp)-mediatedMultidrug Resistance (MDR); 2.5. GSK3 Inhibitors Activities for Substituted imidazoles; 2.6. Anti-inflammatory Activity for Substituted imidazole Derivatives; 2.7. Antimicrobial Activity of Substituted imidazoles i.e. Antibacterial & Antifungal Activity |
|
2.8. Other Biological Activity of Substituted imidazoles3. Methods of Synthesisfor Substituted Imidazoles; Conclusion; References; Chapter 5: Synthesis and Biological Activity of Five-, Six- and Seven-membered S, N-Containing Saturated Heterocycles; Abstract; 1. Introduction; 2. Discussion; 2.1. One-pot Cyclothiomethylation Reaction; 2.2. Biological Activity; Conclusion; References; Chapter 6: Synthesis and Bioactivity of Dihydropyrimidines; Abstract; 1. Introduction; 2. Biological Activities of DHPMs; 2.1. Antifungal Activity; 2.2. Antibacterial Activity; 2.3. Anti-inflammatory Activity |
| Bibliography |
Includes bibliographical references and index |
| Notes |
Print version record |
| Subject |
Heterocyclic compounds -- Synthesis
|
|
Bioactive compounds -- Synthesis
|
|
SCIENCE -- Chemistry -- Organic.
|
|
Heterocyclic compounds -- Synthesis
|
| Form |
Electronic book
|
| Author |
Ameta, K. L., editor
|
|
Pawar, R. P., editor
|
|
Domb, A. J. (Abraham J.), editor.
|
| LC no. |
2019725063 |
| ISBN |
9781622574513 |
|
1622574516 |
|
