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Title Protein kinases as drug targets / edited by Bert Klebl, Gerhard Müller, and Michael Hamacher
Published Weinheim : Wiley-VCH ; Chichester : John Wiley [distributor], [2011]
©2011
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Description 1 online resource (xxi, 373 pages) : illustrations (some color) ; 25 cm
Series Methods and principles in medicinal chemistry ; 49
Methods and principles in medicinal chemistry ; 49
Contents In vitro characterization of small-molecule kinase inhibitors -- Screening for kinase inhibitors: from biochemical to cellular assays -- Dissecting phosphorylation networks: the use of analogue-sensitive kinases and more specific kinase inhibitors as tools -- Rational drug design of kinase inhibitors for signal transduction therapy -- Kinaes inhibitors in signal transduction therapy -- Design principles of deep pocket-targeting protein kinase inhibitors -- From discovery to clinic: aurora kinase inhibitors as novel treatments for cancer -- Discovery and design of protein kinase inhibitors: targeting the cell cycle in oncology -- Medicinal chemistry approaches for the inhibition of the p38 MAPK pathway -- Cellular protein kinases as antiviral targets -- Prospects for TB therapeutics targeting mycobacterium tuberculosis phosphosignaling networks
Bibliography Includes bibliographical references and index
Subject Antineoplastic agents -- Development.
Protein kinases -- Inhibitors.
Protein Kinase Inhibitors -- therapeutic use.
Drug Delivery Systems.
Drug Discovery.
Form Electronic book
Author Klebl, Bert.
Müller, Gerhard, 1963-
Wiley InterScience (Online service)
ISBN 3527633472 (electronic bk.)
3527633480 (electronic bk.)
9783527633470 (electronic bk.)
9783527633487 (electronic bk.)